4-Chloro-3-iodopyridin-2-amine → HCID 58168205, compound

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Reaction Steps

The title compound was synthesized according to the procedure described for the preparation of Example 1 using 4-chloro-3-iodopyridin-2-amine (65 mg, 0.26 mmol) and 5-(2-morpholin-4-yl-ethoxy)-2-(4,4,5,5-tetramethyl[1,3,2]-dioxaborolan-2-yl)-benzoic acid methyl ester (110 mg, 0.28 mmol) to provide 222 (6 mg, 6% yield) as a white solid. LC-MS (M+H=360, obsd.=360).

Provenance & Evidence