Aniline → HCID 58168119, compound

HRID 1029248Notes

Reaction equation

HRID 1029248 reaction equation
F[C:2]1[CH:3]=[C:4]([NH:9][C:10](=[O:33])[CH2:11][C:12]2[NH:16][N:15]=[C:14]([NH:17][C:18]3[CH:27]=[CH:26][N:25]=[C:24]4[C:19]=3[C:20]3[CH:32]=[CH:31][CH:30]=[CH:29][C:21]=3[C:22](=[O:28])[NH:23]4)[CH:13]=2)[CH:5]=[CH:6][C:7]=1F.NC1C=CC=CC=1>>[O:28]=[C:22]1[C:21]2[CH:29]=[CH:30][CH:31]=[CH:32][C:20]=2[C:19]2[C:24](=[N:25][CH:26]=[CH:27][C:18]=2[NH:17][C:14]2[CH:13]=[C:12]([CH2:11][C:10]([NH:9][C:4]3[CH:3]=[CH:2][CH:7]=[CH:6][CH:5]=3)=[O:33])[NH:16][N:15]=2)[NH:23]1

Participants

3

Reactant 2

HCID 6115AnilineHCID 58168312HCID 58168312, compound

Product 1

HCID 58168119HCID 58168119, compound

Procedure

The title compound was synthesized according to the procedure described for the preparation of Example 300 using the carboxylic acid intermediate from example 313 and aniline to provide 315. LC-MS (M+H=411, obsd.=411).

Workup

  1. customThe title compound was synthesized

Sources & evidence

ORD record
ord-341754edbe0945c7a3e10c2d23c7442f
Source dataset
uspto-grants-2014_05
Patent number
US08735584B2

Reaction notes

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