5-Bromopyrimidine-2-carboxylic acid → HCID 67019793, compound

Participants

Reaction Steps

5-(4-((S)-1-((S)-6-(2-hydroxy-2-methylpropyl)-6-isopropyl-2-oxo-1,3-oxazinan-3-yl)ethyl)phenyl)pyrimidine-2-carboxylic acid was prepared from (S)-6-(2-hydroxy-2-methylpropyl)-6-isopropyl-3-((S)-1-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)ethyl)-1,3-oxazinan-2-one and 5-bromopyrimidine-2-carboxylic acid following a procedure analogous to that described in Example 1 Step 2.

Provenance & Evidence