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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1057873Generated: October 26, 2026

Benzylamine → (+/-)-3-(Benzylaminocarbonyl)methyl-4-[(3,5-dichloro-4-pyridyl)aminocarbonyl]-7-methoxy-2,3-dihydrobenzofuran

https://huagongshe.com/reaction/1057873

Reaction equation

Participants

RoleNameHCIDCharge
ReactantBenzylamineHCID 7504—
Reactant(+/-)-3-Carboxymethyl-4-(3,5-dichloro-4-pyridylamino-carbonyl)-7-methoxy-2,3-dihydrobenzofuranHCID 22734342—
Product(+/-)-3-(Benzylaminocarbonyl)methyl-4-[(3,5-dichloro-4-pyridyl)aminocarbonyl]-7-methoxy-2,3-dihydrobenzofuranHCID 2273431565%

Reaction Steps

Substantially the same procedure as in Example 13 was repeated using Compound 9 (0.10 g) obtained in Example 9 and benzylamine to give Compound 25 (0.08 g, 65%) as a white solid.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS06514996B2
Source datasetuspto-grants-2003_02
ORD IDord-d6def2c1dcbe4cb5b731ee6ee8875b97
Source noteuspto-grants-2003_02