Benzylamine → 4-Benzylamino-5-methylsulfonyl-2-methylbenzoic acid

HRID 1058129Notes

Reaction equation

HRID 1058129 reaction equation
[CH3:1][C:2]1[CH:10]=[C:9](Cl)[C:8]([S:12]([CH3:15])(=[O:14])=[O:13])=[CH:7][C:3]=1[C:4]([OH:6])=[O:5].[CH2:16]([NH2:23])[C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1>>[CH2:16]([NH:23][C:9]1[C:8]([S:12]([CH3:15])(=[O:14])=[O:13])=[CH:7][C:3]([C:4]([OH:6])=[O:5])=[C:2]([CH3:1])[CH:10]=1)[C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1

Participants

3

Reactant 2

HCID 7504BenzylamineHCID 108244784-chloro-2-methyl-5-(methylsulfonyl)Benzoic acid

Product 1

HCID 107818944-Benzylamino-5-methylsulfonyl-2-methylbenzoic acid

Procedure

in stage c) 2-methyl-4-chloro-5-methylsulfonylbenzoic acid is reacted with benzylamine to give 4-benzylamino-5-methylsulfonyl-2-methylbenzoic acid,

Sources & evidence

ORD record
ord-d6371f73b5924285ad6305e7f532d20c
Source dataset
uspto-grants-2003_02
Patent number
US06515143B2

Reaction notes

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