Benzylamine → HCID 178454202, compound

HRID 1066745Notes

Reaction equation

[CH2:1]([NH2:8])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.[NH:9]([C:25]([O:27][C:28]([CH3:31])([CH3:30])[CH3:29])=[O:26])[C@H:10]([C:22](O)=[O:23])[CH2:11][CH2:12][CH2:13][NH:14][C:15](=[NH:21])[N:16]([OH:20])[N+:17]([O-:19])=[O:18]>>[NH:9]([C:25]([O:27][C:28]([CH3:31])([CH3:30])[CH3:29])=[O:26])[C@H:10]([C:22]([NH:8][CH2:1][C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1)=[O:23])[CH2:11][CH2:12][CH2:13][NH:14][C:15](=[NH:21])[N:16]([OH:20])[N+:17]([O-:19])=[O:18]

Participants

Reactant 2

HCID 7504Benzylamine

HCID 178454203HCID 178454203, compound

Product 1

HCID 178454202HCID 178454202, compoundYield 81%

Procedure

Boc-Arg(NO2)(OH)CONHBn was prepared according to Example 42 by coupling benzylamine to Boc-Arg(NO2)(OH)COOH in a 81% yield.

Sources & evidence

ORD record: ord-38c97ee4f0454656ae2617960d98313c
Source dataset: uspto-grants-2001_06
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US06245743B1

Reaction notes

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