HCID 15087391, compound → HCID 15087390, compound

HRID 1073684Notes

Reaction equation

HRID 1073684 reaction equation
[C:1]([O:5][C:6]([NH:8][CH2:9][CH2:10][S:11][C:12]1[S:13][CH:14]=[C:15]([C:17]([NH:19][C:20]2[S:21][C:22]3[CH:28]=[CH:27][C:26](F)=[CH:25][C:23]=3[N:24]=2)=[O:18])[N:16]=1)=[O:7])([CH3:4])([CH3:3])[CH3:2].C(OC(NCCSC1SC=C(C(NC2N(C)[C:52]3[CH:55]=[C:56](F)[CH:57]=[CH:58][C:51]=3S2)=O)N=1)=O)(C)(C)C>>[C:1]([O:5][C:6]([NH:8][CH2:9][CH2:10][S:11][C:12]1[S:13][CH:14]=[C:15]([C:17]([NH:19][C:20]2[S:21][C:22]3[CH:28]=[C:27]([C:51]4[CH:58]=[CH:57][CH:56]=[CH:55][CH:52]=4)[CH:26]=[CH:25][C:23]=3[N:24]=2)=[O:18])[N:16]=1)=[O:7])([CH3:4])([CH3:3])[CH3:2]

Participants

3

Reactant 2

HCID 15087391HCID 15087391, compoundHCID 53653837HCID 53653837, compound

Product 1

HCID 15087390HCID 15087390, compound

Procedure

In a similar manner were prepared: 2-(t-butoxy-carbonylaminoethylthio) -N-(5-fluorobenzothiazol-2-yl) -thiazole-4-carboxamide, m.p. 198-199° C. and 2-(t-butoxy-carbonylaminoethylthio)-N-(3-methyl-5-fluorobenzothiazol-2-yl) thiazole-4-carboxamide, m.p. 204-205° C.

Workup

  1. customIn a similar manner were prepared

Sources & evidence

ORD record
ord-5e1196dbfb314292b45d9f0b9691085d
Source dataset
uspto-grants-1990_11
Patent number
US04970318

Reaction notes

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