Boronic Acid → HCID 178440403, compound

HRID 1091924Notes

Reaction equation

HRID 1091924 reaction equation
Br[C:2]1[CH:10]=[CH:9][CH:8]=[C:7]2[C:3]=1[C:4]([CH:11]([CH3:13])[CH3:12])=[N:5][NH:6]2.[BH:14]([OH:16])[OH:15]>>[CH:11]([C:4]1[C:3]2[C:2]([B:14]([OH:16])[OH:15])=[CH:10][CH:9]=[CH:8][C:7]=2[NH:6][N:5]=1)([CH3:13])[CH3:12]

Participants

3

Reactant 2

HCID 61668Boronic AcidHCID 1784404044-Bromo-3-isopropyl-1H-indazole

Product 1

HCID 178440403HCID 178440403, compound

Procedure

4-Bromo-3-isopropyl-1H-indazole is converted to the corresponding boronic acid following analogous procedures to that given in the preceding example. 1H NMR (CD3OD) 7.44(d, 1H), 7.32 (t, 1H), 7.05 (d, 1H), 3.56 (m, 1H), 1.38 (d, 6H). LCMS (m/z): 205.45 (MH)+.

Sources & evidence

ORD record
ord-df74051714954fec8ee927e530f45435
Source dataset
uspto-grants-2012_03
Patent number
US08129395B2

Reaction notes

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