Imidazo[1,2-a]pyridin-3-ylboronic acid → HCID 66592584, compound
Reaction equation
Br[C:2]1[CH:3]=[C:4]([NH:8][C:9]2[CH:13]=[CH:12][O:11][N:10]=2)[CH:5]=[CH:6][CH:7]=1.[N:14]1[CH:15]=[C:16](B(O)O)[N:17]2[CH:22]=[CH:21][CH:20]=[CH:19][C:18]=12>>[N:14]1[CH:15]=[C:16]([C:2]2[CH:3]=[C:4]([NH:8][C:9]3[CH:13]=[CH:12][O:11][N:10]=3)[CH:5]=[CH:6][CH:7]=2)[N:17]2[CH:22]=[CH:21][CH:20]=[CH:19][C:18]=12Participants
3
Procedure
Prepared using procedure outlined in Procedure H using (3-Bromo-phenyl)-isoxazol-3-yl-amine and imidazo[1,2-a]pyridine-3-ylboronic acid as the coupling partners.
Workup
- customPrepared
Sources & evidence
- ORD record
- ord-1eaec7ad031e472fa2e37e23284d3d8e
- Source dataset
- uspto-grants-2012_03
- Patent number
- US08131527B1
Reaction notes
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