HCID 20562695, compound → HCID 54057555, compound

HRID 1155072Notes

Reaction equation

HRID 1155072 reaction equation
Cl.[NH2:2][C:3]1[C:8]([NH2:9])=[CH:7][N:6]=[CH:5][N:4]=1.[CH2:10]([O:13][C:14]1[CH:22]=[C:21]([O:23][CH3:24])[CH:20]=[CH:19][C:15]=1[C:16](Cl)=[O:17])[CH2:11][CH3:12]>>[NH2:2][C:3]1[C:8]([NH:9][C:16](=[O:17])[C:15]2[CH:19]=[CH:20][C:21]([O:23][CH3:24])=[CH:22][C:14]=2[O:13][CH2:10][CH2:11][CH3:12])=[CH:7][N:6]=[CH:5][N:4]=1

Participants

3

Reactant 2

HCID 20562695HCID 20562695, compoundHCID 20562705Pyrimidine-4,5-diamine--hydrogen chloride (1/1)

Product 1

HCID 54057555HCID 54057555, compound

Procedure

The above compound was prepared from 4.4 g of 4,5-diaminopyrimidine hydrochloride and 7.6 g of 2-n-propyloxy-4-methoxy-benzoylchloride using a procedure analogous to that of Example 11(a). The crude product obtained was used in the next step without further purification.

Sources & evidence

ORD record
ord-cd1020658f334847a39fc045ee57d4ec
Source dataset
uspto-grants-1981_11
Patent number
US04299834

Reaction notes

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