HuagongsheHuagongshe Chemistry Print Report · For research reference only
4-Acetylphenylboronic acid → 3-{4-[1-(4'-Acetyl-biphenyl-4-yloxy)-butyl]-benzoylamino}-propionic acid
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 4-Acetylphenylboronic acid | HCID 3702122 | — |
| Reactant | 3-{4-[1-(4-Bromo-phenoxy)-butyl]-benzoylamino}-propionic acid methyl ester | HCID 67153554 | — |
| Product | 3-{4-[1-(4'-Acetyl-biphenyl-4-yloxy)-butyl]-benzoylamino}-propionic acid | HCID 59518156 | — |
Reaction Steps
This compound is made in a substantially similar manner as Example 117 using isomer 1 of 3-{4-[1-(4-bromo-phenoxy)-butyl]-benzoylamino}-propionic acid methyl ester and 4-acetylphenylboronic acid as starting materials in step D. MS (ES): 458.3 [M−H]−.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07816557B2 |
| Source dataset | uspto-grants-2010_10 |
| ORD ID | ord-3cce8099bd7746df881d8cbfae5d9005 |
| Source note | uspto-grants-2010_10 |