(2R,3R,4R,5S)-4,5-bis(Acetoxy)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)tetrahydro-3-furanyl Acetate → (2R,3R,4R,5R)-4-(Acetyloxy)-2-(6-[(2,2-diphenylethyl)amino]-2-{[(isobutylsulphonyl)amino]methyl}9H-purin-9-yl)-5-(5-ethyl-1,2,4-oxadiazol-3-yl)tetrahydro-3-furanyl acetate

Participants

Reaction Steps

Prepared by the same method as Preparation 26 from N-({6-[(2,2-diphenylethyl)amino]-9H-purin-2-yl}methyl)-2-methyl-1-propanesulphonamide hydrochloride (Preparation 8) and (2R,3R,4R,5S)-4,5-bis(acetoxy)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)tetrahydro-3-furanyl acetate (Preparation 38).

Provenance & Evidence