HuagongsheHuagongshe Chemistry Print Report · For research reference only
Benzo[b]furan-2-boronic acid → HCID 9978542, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Benzo[b]furan-2-boronic acid | HCID 2776266 | — |
| Reactant | 2-[3-(3-Chloro-4-fluorophenyl)-8-fluoroimidazo[1,2-alpha]pyridin-7-yl]propan-2-ol | HCID 67486680 | — |
| Product | HCID 9978542 | HCID 9978542 | 3% |
Reaction Steps
2-[3-(3-Chloro-4-fluorophenyl)-8-fluoroimidazo[1,2-α]pyridin-7-yl]-propan-2-ol and benzofuran-2-boronic acid were coupled in the same way as in Example 30 to give 2-{3-[3-(benzofuran-2-yl)-4-fluorophenyl]-8-fluoroimidazo[1,2-α]pyridin-7-yl}propan-2-ol as an off-white solid (6 mg, 3%): m/z (ES+) 405 [MH+].
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07279580B2 |
| Source dataset | uspto-grants-2007_10 |
| ORD ID | ord-708e5f1427354bd1b9387c0188baa157 |
| Source note | uspto-grants-2007_10 |