4-[(Methylsulfonyl)methyl]phenylboronic acid → 4-[5-(4-Methanesulfonylmethylphenyl)-2,3-dihydrofuro[2,3-c]pyridin-2-yl]-piperidine-1-carboxylic acid tert-butyl ester

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Reaction Steps

The title compound is prepared from 4-(5-chloro-2,3-dihydro-furo[2,3-c]pyridin-2-yl)-piperidine-1-carboxylic acid tert-butyl ester and [4-[(methylsulfonyl)methyl]phenyl]boronic acid following a procedure analogous to that described in Example 28. LC (method 10): tR=1.60 min; Mass spectrum (ESI+): m/z=473 [M+H]+.

Provenance & Evidence