HRID1186191
反应详情
EQUATION
反应方程式
REACTANTS
反应物
PRODUCTS
生成物
PROCEDURE
实验过程
The coupling of (R)-5-(5-amino-2-fluorophenyl)-6,6-difluoro-5-methyl-2,5,6,7-tetrahydro-1,4-oxazepin-3-amine (intermediate A10A) and 5-difluoromethoxy-pyridine-2-carboxylic acid (prepared according to Y. Suzuki et al., Int. Patent Appl. No. WO2009091016) yielded the title compound as a pale yellow solid. MS (ISP): m/z=545.2 [M+H]+.