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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1190472Generated: October 27, 2026

2-(4-Methylpiperazino)pyrimidine-5-boronic acid pinacol ester → HCID 58203981, compound

https://huagongshe.com/reaction/1190472

Reaction equation

Participants

RoleNameHCIDCharge
Reactant2-(4-Methylpiperazino)pyrimidine-5-boronic acid pinacol esterHCID 16414228—
Reactant8-Bromo-4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulene-2-carboxylic acid (2-hydroxyethyl)-isopropylamideHCID 67050601—
ProductHCID 58203981HCID 58203981—

Reaction Steps

Following Example 267, 8-Bromo-4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulene-2-carboxylic acid (2-hydroxyethyl)-isopropylamide and 2-(4-methylpiperazin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidine to give 270. MS: (ESI+)=509.2

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08673952B2
Source datasetuspto-grants-2014_03
ORD IDord-6993a984833d4ad2b354f5d964a15142
Source noteuspto-grants-2014_03