4-Formylphenylboronic Acid → HCID 57824419, compound

HRID 1192801Notes

Reaction equation

HRID 1192801 reaction equation
Br[C:2]1[CH:3]=[N:4][CH:5]=[C:6]([C:8]2[CH:13]=[CH:12][C:11]([O:14][C:15]([F:18])([F:17])[F:16])=[CH:10][CH:9]=2)[CH:7]=1.[CH:19]([C:21]1[CH:26]=[CH:25][C:24](B(O)O)=[CH:23][CH:22]=1)=[O:20]>[Pd]>[F:16][C:15]([F:18])([F:17])[O:14][C:11]1[CH:12]=[CH:13][C:8]([C:6]2[CH:7]=[C:2]([C:24]3[CH:25]=[CH:26][C:21]([CH:19]=[O:20])=[CH:22][CH:23]=3)[CH:3]=[N:4][CH:5]=2)=[CH:9][CH:10]=1

Participants

4

Reactant 2

HCID 5910734-Formylphenylboronic AcidHCID 57824470HCID 57824470, compound

Product 1

HCID 57824419HCID 57824419, compound

Reagents, catalysts & solvents 1

HCID 23938PalladiumCatalyst

Procedure

The compound was prepared by palladium-catalyzed arylation of the product of step 1 with 4-formylphenyl boronic acid.

Sources & evidence

ORD record
ord-9bf0c0fd825a40d7beecbb9ae79a5f8c
Source dataset
uspto-grants-2014_03
Patent number
US08680269B2

Reaction notes

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