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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1198965Generated: October 30, 2026

Benzenesulfonamide → N-[4-[6-(N-Cyclopentylmethylcarbamoyl)-3-[2-(morpholinocarbonyl)ethyl]indol-1-ylmethyl]-3-methyoxybenzoyl]benzenesulfonamide

https://huagongshe.com/reaction/1198965

Reaction equation

Participants

RoleNameHCIDCharge
ReactantBenzenesulfonamideHCID 7370—
Reactant4-[6-(N-cyclopentylmethylcarbamoyl)-3-[2-(morpholinocarbonyl)ethyl]indol-1-ylmethyl]-3-methoxybenzoic acidHCID 15013781—
ProductN-[4-[6-(N-Cyclopentylmethylcarbamoyl)-3-[2-(morpholinocarbonyl)ethyl]indol-1-ylmethyl]-3-methyoxybenzoyl]benzenesulfonamideHCID 19867561—

Reaction Steps

Using a similar procedure to the described in Example 2, but starting from 4-[6-(N-cyclopentylmethylcarbamoyl)-3-[2-(morpholinocarbonyl)ethyl]indol-1-ylmethyl]-3-methoxybenzoic acid and phenylsulfonamide, the title compound was obtained as a white solid (69%); mp 244°-245°.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS04898863
Source datasetuspto-grants-1990_02
ORD IDord-1eb1cd984ac847f0a5911b7a8c6ae547
Source noteuspto-grants-1990_02