5-(1-Phenylethyl)benzofuran-2-ylboronic acid → Methyl 1-((3-fluoro-4-(5-(1-phenylethyl)benzofuran-2-yl)phenyl)methyl)azetidine-3-carboxylate
Reaction equation
[Br:1][c:2]1[c:3]([F:17])[cH:4][c:5]([CH2:6][N:7]2[CH2:8][CH:9]([C:11](=[O:12])[O:13][CH3:14])[CH2:10]2)[cH:15][cH:16]1.[c:18]1([CH:24]([CH3:25])[c:26]2[cH:27][cH:28][c:29]3[c:30]([cH:31][c:32]([B:34]([OH:35])[OH:36])[o:33]3)[cH:37]2)[cH:19][cH:20][cH:21][cH:22][cH:23]1>>[c:2]1(-[c:32]2[cH:31][c:30]3[c:29]([cH:28][cH:27][c:26]([CH:24]([c:18]4[cH:19][cH:20][cH:21][cH:22][cH:23]4)[CH3:25])[cH:37]3)[o:33]2)[c:3]([F:17])[cH:4][c:5]([CH2:6][N:7]2[CH2:8][CH:9]([C:11](=[O:12])[O:13][CH3:14])[CH2:10]2)[cH:15][cH:16]1Participants
3
Sources & evidence
- ORD record
- ord-c7fa6fcb80174b9a8077e62d3b24f7dc
- Source dataset
- Training data from https://doi.org/10.1039/C8SC04228D (5/10)
Reaction notes
Loading…