HuagongsheHuagongshe Chemistry Print Report · For research reference only
2-Methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenol → 4-{6-[(2-Furylmethyl)amino]pyrazin-2-yl}-2-methoxyphenol
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 2-Methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenol | HCID 2734650 | — |
| Reactant | N-(6-Chloro-2-pyrazinyl)-N-(2-furylmethyl)amine | HCID 21919348 | — |
| Product | 4-{6-[(2-Furylmethyl)amino]pyrazin-2-yl}-2-methoxyphenol | HCID 135516741 | 92% |
Reaction Steps
In a procedure analogous to Example 2, reaction of 6-chloro-N-(2-furylmethyl)pyrazin-2-amine and 2-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenol furnished the product (92%).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07122550B2 |
| Source dataset | uspto-grants-2006_10 |
| ORD ID | ord-e5ba14bdf822409aba7beae794f93e9c |
| Source note | uspto-grants-2006_10 |