Cyclopropanemethanamine → HCID 57377807, compound

Participants

Reaction Steps

As described for example 43c, 6-(4-(1-(2-fluorophenyl)-4-methyl-1H-1,2,3-triazol-5-yl)-1H-imidazol-1-yl)nicotinic acid (74 mg, 0.203 mmol) was converted, using aminomethylcyclopropane instead of isopropylamine, to the title compound (40 mg, 47%) which was obtained as a white foam after purification by chromatography (reverse phase HPLC). MS: m/e=418.3 [M+H]+.

Provenance & Evidence