4-Quinolinecarboxylic acid → HCID 178523738, compound

Participants

Reaction Steps

The title compound, white solid (80 mg, 66%), MS (ISP) m/z=486.6 [(M+H)+], mp 222° C., was prepared in accordance with the general method of example 6 from trans-4-{2-[4-(2,3-dihydro-furo[2,3-c]pyridin-7-yl)-piperazin-1-yl]-ethyl}-cyclohexylamine trihydrochloride (intermediate B) (110 mg, 0.25 mmol) and quinoline-4-carboxylic acid.

Provenance & Evidence