Racemic trans-(3-methoxy-cyclopentyl)-acetic acid methyl ester → HCID 178496553, compound

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Reaction Steps

The title compound, white solid (117 mg, 99%), MS (ISP) m/z=471.6 [(M+H)+], mp 199° C., was prepared in accordance with the general method of example 5 from trans-4-{2-[4-(2,3-dihydro-furo[2,3-c]pyridin-7-yl)-piperazin-1-yl]-ethyl}-cyclohexylamine trihydrochloride (intermediate B) (110 mg, 0.25 mmol) and methyl 2-((1S,3S)-3-methoxy-cyclopentyl)-acetate.

Provenance & Evidence