3-(5-Methyl-1,2,4-oxadiazol-3-yl)benzoic acid → HCID 178432504, compound

Participants

Reaction Steps

The title compound, white solid (120 mg, 93%), MS (ISP) m/z=517.5 [(M+H)+], mp 227.5° C., was prepared in accordance with the general method of example 6 from trans-4-{2-[4-(2,3-dihydro-furo[2,3-c]pyridin-7-yl)-piperazin-1-yl]-ethyl}-cyclohexylamine trihydrochloride (intermediate B) (110 mg, 0.25 mmol) and 3-(5-methyl-[1,2,4]oxadiazol-3-yl)-benzoic acid.

Provenance & Evidence