Ethylamine → HCID 178514748, compound
Reaction equation
FC1C(O[C:9]([C:11]2[CH:12]=[C:13]3[C:17](=[CH:18][CH:19]=2)[NH:16][C:15](=[O:20])[C:14]3=[N:21][NH:22][C:23]2[CH:28]=[CH:27][C:26]([S:29](=[O:32])(=[O:31])[NH2:30])=[CH:25][CH:24]=2)=[O:10])=C(F)C(F)=C(F)C=1F.[CH2:37]([NH2:39])[CH3:38]>>[N:39]1([CH2:14][CH2:15][NH:16][C:9]([C:11]2[CH:12]=[C:13]3[C:17](=[CH:18][CH:19]=2)[NH:16][C:15](=[O:20])[C:14]3=[N:21][NH:22][C:23]2[CH:24]=[CH:25][C:26]([S:29](=[O:32])(=[O:31])[NH2:30])=[CH:27][CH:28]=2)=[O:10])[CH2:11][CH2:9][O:10][CH2:38][CH2:37]1Participants
3
Procedure
The title compound was prepared from 2-oxo-3[(4-sulfamoyl-phenyl)-hydrazono]-2,3-dihydro-1H-indole-5-carboxylic acid pentafluorophenyl ester and 2-N-morpholino)ethylamine according to Procedure K: mp210-212° C.; Anal. Calcd for C21H24N6O5S.1/4H2O: C, 52.88; H, 5.18; N, 17.62. Found: C, 52.91; H, 5.24; N, 17.35.
Sources & evidence
- ORD record
- ord-a809ca36d6eb4caeb2dce478a4e0fc6b
- Source dataset
- uspto-grants-2003_04
- Patent number
- US06541503B2
Reaction notes
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