1-Deoxy-1-(methylamino)-D-galactitol → N-[2-(3-Cyano-1H-indol-5-yl)-ethyl]-4-{2-[methyl-(2 (S),3 (R),4 (S),5 (R),6-pentahydroxy-hexyl)-amino]-pyrimidin-4-yl}-benzamide

Participants

Role	Name	HCID	Charge
Reactant	1-Deoxy-1-(methylamino)-D-galactitol	HCID 12598090	—
Reactant	N-[2-(3-Cyano-1H-indol-5-yl)-ethyl]-4-[2-chloropyrimidin-4-yl]benzamide	HCID 18617562	—
Product	N-[2-(3-Cyano-1H-indol-5-yl)-ethyl]-4-{2-[methyl-(2 (S),3 (R),4 (S),5 (R),6-pentahydroxy-hexyl)-amino]-pyrimidin-4-yl}-benzamide	HCID 70030820	—

Reaction Steps

Using N-methyl-(2 (S),3 (R),4 (S),5 (R),6-pentahydroxy-hexyl)-amine and N-[2-(3-Cyano-1H-indol-5-yl)-ethyl]-4-[2-chloro-pyrimidin-4-yl]-benzamide (reference example 1az) as substrates.

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US06541505B1
Source dataset	uspto-grants-2003_04
ORD ID	ord-1cf5838aef674d65abdc0fdefa73a66a
Source note	uspto-grants-2003_04