Tolylboronic acid → HCID 16125882, compound

HRID 1267632Notes

Reaction equation

HRID 1267632 reaction equation
[CH3:1][C:2]1[CH:7]=[CH:6][C:5](B(O)O)=[CH:4][CH:3]=1.Cl[C:12]1[CH:13]=[C:14]([CH:20]=[CH:21][N:22]=1)[C:15]([O:17][CH2:18][CH3:19])=[O:16]>>[CH3:1][C:2]1[CH:7]=[CH:6][C:5]([C:12]2[CH:13]=[C:14]([CH:20]=[CH:21][N:22]=2)[C:15]([O:17][CH2:18][CH3:19])=[O:16])=[CH:4][CH:3]=1

Participants

3

Reactant 2

HCID 79799Tolylboronic acidHCID 2762942Ethyl 2-chloroisonicotinate

Product 1

HCID 16125882HCID 16125882, compound

Procedure

4-Methylphenylboronic acid (161 mg) and ethyl 2-chloroisonicotinate (200 mg) were treated in the same manner as in Preparation Example 1 to obtain the title compound.

Sources & evidence

ORD record
ord-7a1c24c058d94caa9636c0e000901a36
Source dataset
uspto-grants-2003_04
Patent number
US06552188B2

Reaction notes

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