4-Chlorophenylboronic acid → HCID 18448292, compound

HRID 1269696Notes

Reaction equation

HRID 1269696 reaction equation
[Cl:1][C:2]1[CH:7]=[CH:6][C:5](B(O)O)=[CH:4][CH:3]=1.Br[C:12]1[C:13]([CH3:38])=[C:14]([N:18]([CH2:23][C:24]2[CH:36]=[CH:35][C:27]([O:28][CH2:29][C:30]([O:32]CC)=[O:31])=[C:26]([CH3:37])[CH:25]=2)[CH2:19][CH2:20][O:21][CH3:22])[CH:15]=[CH:16][CH:17]=1>>[Cl:1][C:2]1[CH:7]=[CH:6][C:5]([C:12]2[CH:17]=[CH:16][CH:15]=[C:14]([N:18]([CH2:23][C:24]3[CH:36]=[CH:35][C:27]([O:28][CH2:29][C:30]([OH:32])=[O:31])=[C:26]([CH3:37])[CH:25]=3)[CH2:19][CH2:20][O:21][CH3:22])[C:13]=2[CH3:38])=[CH:4][CH:3]=1

Participants

3

Reactant 2

HCID 742994-Chlorophenylboronic acidHCID 58622864HCID 58622864, compound

Product 1

HCID 18448292HCID 18448292, compound

Procedure

Prepared from 4-chlorophenylboronic acid and ethyl (4-{[(3-bromo-2-methylphenyl)(2-methoxyethyl)amino]methyl}-2-methylphenoxy)acetate using the procedure described for Example 25 (Method A).

Sources & evidence

ORD record
ord-eb746e45621d464bb4d0683ceeab7424
Source dataset
uspto-grants-2007_04
Patent number
US07199239B2

Reaction notes

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