4-Chlorophenylboronic acid → HCID 18448293, compound

HRID 1269699Notes

Reaction equation

HRID 1269699 reaction equation
[Cl:1][C:2]1[CH:7]=[CH:6][C:5](B(O)O)=[CH:4][CH:3]=1.Br[C:12]1[C:13]([CH3:37])=[C:14]([N:18]([CH2:22][C:23]2[CH:35]=[CH:34][C:26]([O:27][CH2:28][C:29]([O:31]CC)=[O:30])=[C:25]([CH3:36])[CH:24]=2)[CH2:19][CH2:20][CH3:21])[CH:15]=[CH:16][CH:17]=1>>[Cl:1][C:2]1[CH:7]=[CH:6][C:5]([C:12]2[CH:17]=[CH:16][CH:15]=[C:14]([N:18]([CH2:22][C:23]3[CH:35]=[CH:34][C:26]([O:27][CH2:28][C:29]([OH:31])=[O:30])=[C:25]([CH3:36])[CH:24]=3)[CH2:19][CH2:20][CH3:21])[C:13]=2[CH3:37])=[CH:4][CH:3]=1

Participants

3

Reactant 2

HCID 742994-Chlorophenylboronic acidHCID 58622881HCID 58622881, compound

Product 1

HCID 18448293HCID 18448293, compound

Procedure

Prepared from 4-chlorophenylboronic acid and ethyl (4-{[(3-bromo-2-methylphenyl)(propyl)amino]methyl}-2-methylphenoxy)acetate using the procedure described Example 25.

Sources & evidence

ORD record
ord-7618e14acf274df6a8e6e9fcdcf8f90a
Source dataset
uspto-grants-2007_04
Patent number
US07199239B2

Reaction notes

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