4-Cyanophenylboronic acid → HCID 18448294, compound

HRID 1269702Notes

Reaction equation

HRID 1269702 reaction equation
[C:1]([C:3]1[CH:8]=[CH:7][C:6](B(O)O)=[CH:5][CH:4]=1)#[N:2].Br[C:13]1[C:14]([CH3:38])=[C:15]([N:19]([CH2:23][C:24]2[CH:36]=[CH:35][C:27]([O:28][CH2:29][C:30]([O:32]CC)=[O:31])=[C:26]([CH3:37])[CH:25]=2)[CH2:20][CH2:21][CH3:22])[CH:16]=[CH:17][CH:18]=1>>[C:1]([C:3]1[CH:8]=[CH:7][C:6]([C:13]2[CH:18]=[CH:17][CH:16]=[C:15]([N:19]([CH2:23][C:24]3[CH:36]=[CH:35][C:27]([O:28][CH2:29][C:30]([OH:32])=[O:31])=[C:26]([CH3:37])[CH:25]=3)[CH2:20][CH2:21][CH3:22])[C:14]=2[CH3:38])=[CH:5][CH:4]=1)#[N:2]

Participants

3

Reactant 2

HCID 27343264-Cyanophenylboronic acidHCID 58622881HCID 58622881, compound

Product 1

HCID 18448294HCID 18448294, compound

Procedure

Prepared from 4-cyanophenylboronic acid and ethyl (4-{[(3-bromo-2-methylphenyl)(propyl)amino]methyl}-2-methylphenoxy)acetate using the procedure described for Example 25 (Method A).

Sources & evidence

ORD record
ord-f6c9f2b5c5564ad39b92b689639aac04
Source dataset
uspto-grants-2007_04
Patent number
US07199239B2

Reaction notes

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