HuagongsheHuagongshe Chemistry Print Report · For research reference only
3-Pyridinylboronic acid → N-[4-Methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-(pyridin-3-yl)naphth-1-ylacetamide
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 3-Pyridinylboronic acid | HCID 2734378 | — |
| Reactant | 4-Bromo-N-[4-methoxy-3-(4-methylpiperizin-1-yl)phenyl]naphth-1-yl Acetamide | HCID 22118888 | — |
| Product | N-[4-Methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-(pyridin-3-yl)naphth-1-ylacetamide | HCID 22118931 | — |
Reaction Steps
The title compound was prepared from 4-bromo-N-[4-methoxy-3-(4-methyipiperazin-1-yl)phenyl]-1-naphthylacetamide (E9) and 3-pyridylboronic acid using a similar procedure to Example 4 as a white solid (32%).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US06159979 |
| Source dataset | uspto-grants-2000_12 |
| ORD ID | ord-acd181a5e1614f2082587609493a7067 |
| Source note | uspto-grants-2000_12 |