1-(Phenylmethyl)-1H-indazol-5-amine → HCID 23589545, compound

HRID 1295762Notes

Reaction equation

HRID 1295762 reaction equation
[CH2:1]([O:3][C:4]([C:6]1[C:7]([CH2:23][CH3:24])=[C:8]2[N:13]([CH:14]=1)[N:12]=[CH:11][N:10]=[C:9]2[NH:15][C:16]1[CH:21]=[CH:20][C:19](Br)=[CH:18][CH:17]=1)=[O:5])[CH3:2].NC1C=C2C(=CC=1)[N:31]([CH2:35][C:36]1[CH:41]=[CH:40][CH:39]=[CH:38][CH:37]=1)[N:30]=[CH:29]2>>[CH2:1]([O:3][C:4]([C:6]1[C:7]([CH2:23][CH3:24])=[C:8]2[N:13]([CH:14]=1)[N:12]=[CH:11][N:10]=[C:9]2[NH:15][C:16]1[CH:21]=[C:20]2[C:19](=[CH:18][CH:17]=1)[N:31]([CH2:35][C:36]1[CH:41]=[CH:40][CH:39]=[CH:38][CH:37]=1)[N:30]=[CH:29]2)=[O:5])[CH3:2]

Participants

3

Reactant 2

HCID 2120691-(Phenylmethyl)-1H-indazol-5-amineHCID 23589547HCID 23589547, compound

Product 1

HCID 23589545HCID 23589545, compound

Procedure

The title compound was prepared from compound B of Example 139 using the process described for the preparation of example 139 except 5-amino-1-benzyl-1H-indazole was used to add to the chloroimidate. MS: (M+H)+=441.24

Sources & evidence

ORD record
ord-947e2932c8414e30bf3127f91dff4b02
Source dataset
uspto-grants-2007_07
Patent number
US07244733B2

Reaction notes

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