Benzyl succinimido carbonate → HCID 10293195, compound

HRID 1351586Notes

Reaction equation

HRID 1351586 reaction equation
[C:1]([C:3]1[N:4]=[C:5]([O:17][CH3:18])[C:6]([NH:9][CH2:10][CH:11]2[CH2:16][CH2:15][NH:14][CH2:13][CH2:12]2)=[N:7][CH:8]=1)#[N:2].[CH2:19]([O:26][C:27](ON1C(=O)CCC1=O)=[O:28])[C:20]1[CH:25]=[CH:24][CH:23]=[CH:22][CH:21]=1>>[CH2:19]([O:26][C:27]([N:14]1[CH2:15][CH2:16][CH:11]([CH2:10][NH:9][C:6]2[C:5]([O:17][CH3:18])=[N:4][C:3]([C:1]#[N:2])=[CH:8][N:7]=2)[CH2:12][CH2:13]1)=[O:28])[C:20]1[CH:25]=[CH:24][CH:23]=[CH:22][CH:21]=1

Participants

3

Reactant 2

HCID 83172Benzyl succinimido carbonateHCID 22135674HCID 22135674, compound

Product 1

HCID 10293195HCID 10293195, compound

Procedure

The above compound was prepared in a similar manner as described in EXAMPLE 130 from 4-[(5-cyano-3-methoxy-pyrazin-2-ylamino)-methyl]-piperidine using N-(benzyloxycarbonyloxy)succinimide (Sigma-Aldrich). M.S. (M+1): 382.

Workup

  1. customThe above compound was prepared in a similar manner

Sources & evidence

ORD record
ord-62d664cacd604ab8bd603481f1ef62fc
Source dataset
uspto-grants-2007_05
Patent number
US07217716B2

Reaction notes

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