3-(Phenylsulfonyl)propanoic acid → HCID 57954722, compound

Participants

Reaction Steps

The title compound is prepared analogously as described in example G1 using (S)-2-methyl-propane-2-sulfinic acid [(R)-1-piperidin-4-yl-2-(2,4,5-trifluoro-phenyl)-ethyl]-amide instead of 3-exo-[(R)-1-((S)-2-methyl-propane-2-sulfinylamino)-2-(2,4,5-trifluoro-phenyl)-ethyl]-8-aza-bicyclo[3.2.1]octane and 3-benzenesulfonyl-propionic acid instead of N-acetyl-L-alanine.

Provenance & Evidence