(3-Methoxyphenyl)boronic acid → HCID 18512349, compound

HRID 1370823Notes

Reaction equation

HRID 1370823 reaction equation
[F:1][C:2]1[CH:27]=[C:26]([F:28])[CH:25]=[CH:24][C:3]=1[CH2:4][N:5]([CH2:16][C:17]1[CH:22]=[CH:21][C:20]([OH:23])=[CH:19][CH:18]=1)[C:6]1[CH:11]=[CH:10][CH:9]=[C:8]([N+:12]([O-:14])=[O:13])[C:7]=1[CH3:15].[CH3:29][O:30][C:31]1[CH:32]=[C:33](B(O)O)[CH:34]=[CH:35][CH:36]=1>>[F:1][C:2]1[CH:27]=[C:26]([F:28])[CH:25]=[CH:24][C:3]=1[CH2:4][N:5]([CH2:16][C:17]1[CH:22]=[CH:21][C:20]([O:23][C:35]2[CH:34]=[CH:33][CH:32]=[C:31]([O:30][CH3:29])[CH:36]=2)=[CH:19][CH:18]=1)[C:6]1[CH:11]=[CH:10][CH:9]=[C:8]([N+:12]([O-:14])=[O:13])[C:7]=1[CH3:15]

Participants

3

Reactant 2

HCID 2734370(3-Methoxyphenyl)boronic acidHCID 18512160N-(2,4-difluorobenzyl)-N-(4-hydroxybenzyl)-2-methyl-3-nitroaniline

Product 1

HCID 18512349HCID 18512349, compound

Procedure

The product from Example 33A and 3-methoxyphenylboronic acid were processed as described in Example 48A to provide the title compound.

Sources & evidence

ORD record
ord-616d6feed8c3467da0734d8690ea4847
Source dataset
uspto-grants-2003_06
Patent number
US06583180B2

Reaction notes

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