反应详情

In an analogous manner to that described in Example 20 d), the condensation of (S)-3-amino-5-(2,2-dimethyl-propionyl)-1-methyl-1,3,4,5-tetrahydro-benzo[b][1,4]diazepin-2-one hydrochloride and N-(2,2,3,3,3-pentafluoro-propyl)-malonamic acid yielded the title compound as a white foam;

1. customdescribed in Example 20 d