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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1379372Generated: October 30, 2026

Carbodiimide → 2-(t-Butyloxycarbonylamino)-4-(N-((p-toluenesulfonyl)valinyl)amino)-1,5-diphenyl-3-hydroxypentane

https://huagongshe.com/reaction/1379372

Reaction equation

Participants

RoleNameHCIDCharge
ReactantCarbodiimideHCID 160435—
ReactantTosyl valineHCID 2249310—
Reactant4-Amino-2-(t-butyloxycarbonylamino)-1,5-diphenyl-3-hydroxypentaneHCID 14704377—
Product2-(t-Butyloxycarbonylamino)-4-(N-((p-toluenesulfonyl)valinyl)amino)-1,5-diphenyl-3-hydroxypentaneHCID 22845645—

Reaction Steps

According to the carbodiimide coupling procedure of Example 55, N-(p-toluenesulfonyl)valine was coupled to the resultant compound of Example 11 to give the desired compound.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS05670675
Source datasetuspto-grants-1997_09
ORD IDord-0048facf8be6489992a8e94709d922a6
Source noteuspto-grants-1997_09