HCID 15545704, compound → HCID 21716365, compound

HRID 1385904Notes

Reaction equation

HRID 1385904 reaction equation
[CH3:1][O:2][C:3]1[CH:4]=[C:5]([CH:11]2[O:16][CH2:15][C:14](=[O:17])[NH:13][CH2:12]2)[CH:6]=[CH:7][C:8]=1[O:9][CH3:10].N[CH2:19][CH:20]([C:22]1C=CC(OC)=C(OC2CCCC2)[CH:23]=1)O>>[CH:1]1([O:2][C:3]2[CH:4]=[C:5]([CH:11]3[O:16][CH2:15][C:14](=[O:17])[NH:13][CH2:12]3)[CH:6]=[CH:7][C:8]=2[O:9][CH3:10])[CH2:23][CH2:22][CH2:20][CH2:19]1

Participants

3

Reactant 2

HCID 15545704HCID 15545704, compoundHCID 21716356HCID 21716356, compound

Product 1

HCID 21716365HCID 21716365, compoundYield 42.7%

Procedure

According to the same procedure as in Example 1(2) to (3), using 2-amino-1-(3-cyclopentyloxy-4-methoxyphenyl)ethanol instead of 2-amino-1-(3,4-dimethoxyphenyl)ethanol, the above-described compound (yield 42.7%) was obtained as a colorless solid.

Sources & evidence

ORD record
ord-b44ec0270112457789881efb8e3f52d8
Source dataset
uspto-grants-2001_07
Patent number
US06265402B1

Reaction notes

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