Benzenepropanoyl chloride → HCID 69312997, compound

Participants

Reaction Steps

In accordance with the same procedure as in Example 87, except that 4-[N-[1-[N-(4-fluorobenzoyl)amino]cyclohexanecarbonyl]amino]-1-(4-fluoro-2-aminophenyl)piperidin-3-ol was used instead of 4-[N-[1-[N-(furan-2-ylcarbonyl)amino]cyclohexanecarbonyl]amino]-1-(4-fluoro-2-aminophenyl)piperidin-3-ol and hydrocinnamoyl chloride was used instead of methoxyacetyl chloride in Step 3 thereof, 671 mg of the titled compound was prepared.

Provenance & Evidence