4-Amino-1-Boc-piperidine → HCID 59681751, compound

HRID 1394191Notes

Reaction equation

HRID 1394191 reaction equation
C(OC([N:8]1[CH2:13][CH2:12][CH:11]([NH2:14])[CH2:10][CH2:9]1)=O)(C)(C)C.[NH2:15][C:16]1[C:17]([C:21]2[N:22]([CH2:38][CH3:39])[C:23]3[C:28]([C:29]4[CH:30]=[C:31]([CH:34]=[CH:35][CH:36]=4)[CH:32]=O)=[CH:27][N:26]=[CH:25][C:24]=3[N:37]=2)=[N:18][O:19][N:20]=1>>[NH2:15][C:16]1[C:17]([C:21]2[N:22]([CH2:38][CH3:39])[C:23]3[C:28]([C:29]4[CH:30]=[C:31]([CH:34]=[CH:35][CH:36]=4)[CH2:32][NH:14][CH:11]4[CH2:10][CH2:9][NH:8][CH2:13][CH2:12]4)=[CH:27][N:26]=[CH:25][C:24]=3[N:37]=2)=[N:18][O:19][N:20]=1

Participants

3

Reactant 2

HCID 12682914-Amino-1-Boc-piperidineHCID 131726811HCID 131726811, compound

Product 1

HCID 59681751HCID 59681751, compound

Procedure

The title compound was prepared from 4-amino-piperidine-1-carboxylic acid tert-butyl ester and the product of Example 153 Step 1 using the method of Example 149, followed by the method described in Example 21. MS (ES+) m/e 419 [M+H]+.

Sources & evidence

ORD record
ord-92dfd33cb45745b59391d13a122e2f07
Source dataset
uspto-grants-2008_03
Patent number
US07348339B2

Reaction notes

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