4-Methoxyphenoxyacetic acid → HCID 66758804, compound

HRID 1396773Notes

Reaction equation

HRID 1396773 reaction equation
[CH2:1]([C:6]1[S:7][C:8]2[N:9]=[C:10]([NH2:21])[N:11]=[C:12]([N:15]3[CH2:20][CH2:19][NH:18][CH2:17][CH2:16]3)[C:13]=2[N:14]=1)[CH2:2][CH2:3][CH2:4][CH3:5].[CH3:22][O:23][C:24]1[CH:34]=[CH:33][C:27]([O:28][CH2:29][C:30](O)=[O:31])=[CH:26][CH:25]=1>>[NH2:21][C:10]1[N:11]=[C:12]([N:15]2[CH2:20][CH2:19][N:18]([C:30](=[O:31])[CH2:29][O:28][C:27]3[CH:33]=[CH:34][C:24]([O:23][CH3:22])=[CH:25][CH:26]=3)[CH2:17][CH2:16]2)[C:13]2[N:14]=[C:6]([CH2:1][CH2:2][CH2:3][CH2:4][CH3:5])[S:7][C:8]=2[N:9]=1

Participants

3

Reactant 2

HCID 746494-Methoxyphenoxyacetic acidHCID 50942149HCID 50942149, compound

Product 1

HCID 66758804HCID 66758804, compoundYield 34%

Procedure

This compound was prepared from 2-pentyl-7-(piperazin-1-yl)thiazolo[5,4-d]pyrimidin-5-amine using 4-methoxyphenoxyacetic acid in a yield of 34%, according to the procedure for the synthesis of example 50.

Workup

  1. customaccording to the procedure for the synthesis of example 50

Sources & evidence

ORD record
ord-0a56046b841e412b9ce084ab80908b3f
Source dataset
uspto-grants-2014_12
Patent number
US08901132B2

Reaction notes

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