HuagongsheHuagongshe Chemistry Print Report · For research reference only
3-(2-Dimethylaminoethylaminocarbonyl)benzeneboronic acid → 3-{1-[1-(2,6-dichloro-3-fluorophenyl)ethoxy]-1H-pyrrolo[3,2-b]pyridin-6-yl}-N-[2-(dimethylamino)ethyl]benzamide
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 3-(2-Dimethylaminoethylaminocarbonyl)benzeneboronic acid | HCID 44119531 | — |
| Reactant | 6-bromo-1-[1-(2,6-dichloro-3-fluorophenyl)ethoxy]-1H-pyrrolo[3,2-b]pyridine | HCID 67458418 | — |
| Product | 3-{1-[1-(2,6-dichloro-3-fluorophenyl)ethoxy]-1H-pyrrolo[3,2-b]pyridin-6-yl}-N-[2-(dimethylamino)ethyl]benzamide | HCID 86659798 | — |
Reaction Steps
The entitled compound was prepared from 6-bromo-1-[1-(2,6-dichloro-3-fluorophenyl)ethoxy]-1H-pyrrolo[3,2-b]pyridine and (3-{[2-(dimethylamino)ethyl]carbamoyl}phenyl)boronic acid according to the procedure described in example 4.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08912330B2 |
| Source dataset | uspto-grants-2014_12 |
| ORD ID | ord-499bc06155f14c31b6f5412cc3e1f4c7 |
| Source note | uspto-grants-2014_12 |