(1-Benzofuran-5-yl)boronic acid → HCID 58532432, compound

HRID 1404604Notes

Reaction equation

HRID 1404604 reaction equation
Br[C:2]1[CH:3]=[C:4]2[N:10]([O:11][C:12]3[CH:17]=[CH:16][CH:15]=[CH:14][CH:13]=3)[CH:9]=[CH:8][C:5]2=[N:6][CH:7]=1.[O:18]1[C:22]2[CH:23]=[CH:24][C:25](B(O)O)=[CH:26][C:21]=2[CH:20]=[CH:19]1>>[O:18]1[C:22]2[CH:23]=[CH:24][C:25]([C:2]3[CH:3]=[C:4]4[N:10]([O:11][C:12]5[CH:17]=[CH:16][CH:15]=[CH:14][CH:13]=5)[CH:9]=[CH:8][C:5]4=[N:6][CH:7]=3)=[CH:26][C:21]=2[CH:20]=[CH:19]1

Participants

3

Reactant 2

HCID 4197999(1-Benzofuran-5-yl)boronic acidHCID 58532385HCID 58532385, compound

Product 1

HCID 58532432HCID 58532432, compoundYield 25%

Procedure

The entitled compound was prepared from 6-bromo-1-phenoxy-1H-pyrrolo[3,2-b]pyridine and 1-benzofuran-5-ylboronic acid in a 25% yield according to the procedure described in example 23.

Sources & evidence

ORD record
ord-dbebbd7109ee41dab0832f712bac5c07
Source dataset
uspto-grants-2014_12
Patent number
US08912330B2

Reaction notes

Loading…