HuagongsheHuagongshe Chemistry Print Report · For research reference only
2-Amino-5-fluorobenzoic acid → HCID 86723064, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 2-Amino-5-fluorobenzoic acid | HCID 101412 | — |
| Reactant | 6-[(R)-5-(3-amino-propyl)-2-oxo-oxazolidin-3-yl]-4H-benzo[1,4]thiazin-3-one | HCID 67303587 | — |
| Product | HCID 86723064 | HCID 86723064 | 70% |
Reaction Steps
Starting from 2-amino-5-fluorobenzoic acid and 6-[(R)-5-(3-amino-propyl)-2-oxo-oxazolidin-3-yl]-4H-benzo[1,4]thiazin-3-one (described in WO 2010/041219) and using Procedure D, the title compound was obtained as a beige solid (160 mg; 70% yield).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08916573B2 |
| Source dataset | uspto-grants-2014_12 |
| ORD ID | ord-ddfc193a3a0d4fb8b7089947e336d775 |
| Source note | uspto-grants-2014_12 |