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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1405628Generated: October 30, 2026

4-Fluoroanthranilic acid → HCID 86723066, compound

https://huagongshe.com/reaction/1405628

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-Fluoroanthranilic acidHCID 2724967—
Reactant6-[(R)-5-(3-amino-propyl)-2-oxo-oxazolidin-3-yl]-4H-benzo[1,4]thiazin-3-oneHCID 67303587—
ProductHCID 86723066HCID 8672306678%

Reaction Steps

Starting from 2-amino-4-fluorobenzoic acid and 6-[(R)-5-(3-amino-propyl)-2-oxo-oxazolidin-3-yl]-4H-benzo[1,4]thiazin-3-one (described in WO 2010/041219) and using Procedure D, the title compound was obtained as a beige solid (130 mg; 78% yield).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08916573B2
Source datasetuspto-grants-2014_12
ORD IDord-480bbd2c3c6146ffb96c835f08a6a5e6
Source noteuspto-grants-2014_12