2-Methanesulfonylacetic acid → HCID 178504899, compound

Participants

Reaction Steps

The title compound, white solid (79 mg, 71%), MS (ISP) m/z=447.3 [(M+H)+], mp 187° C., was prepared in accordance with the general method of example 1 from trans-4-[2-(4-benzofuran-3-yl-piperidin-1-yl)-ethyl]-cyclohexylamine dihydrochloride (intermediate A) (100 mg, 0.25 mmol) and 2-methanesulfonyl-acetic acid.

Provenance & Evidence