4-Quinolinecarboxylic acid → HCID 178523656, compound

Participants

Reaction Steps

The title compound, yellow solid (106 mg, 88%), MS (ISP) m/z=482.3 [(M+H)+], mp 169° C., was prepared in accordance with the general method of example 1 from trans-4-[2-(4-benzofuran-3-yl-piperidin-1-yl)-ethyl]-cyclohexylamine dihydrochloride (intermediate A) (100 mg, 0.25 mmol) and quinoline-4-carboxylic acid.

Provenance & Evidence