3-Hydroxypropionic acid → HCID 178520898, compound

Participants

Reaction Steps

The title compound, off-white solid (20 mg, 20%), MS (ISP) m/z=399.3 [(M+H)+], mp 148° C., was prepared in accordance with the general method of example 1 from trans-4-[2-(4-benzofuran-3-yl-piperidin-1-yl)-ethyl]-cyclohexylamine dihydrochloride (intermediate A) (100 mg, 0.25 mmol) and 3-hydroxy-propionic acid.

Provenance & Evidence