6-Methylnicotinic acid → HCID 178425860, compound

Participants

Reaction Steps

The title compound, yellow solid (66 mg, 59%), MS (ISP) m/z=446.4 [(M+H)+], mp 203° C., was prepared in accordance with the general method of example 1 from trans-4-[2-(4-benzofuran-3-yl-piperidin-1-yl)-ethyl]-cyclohexylamine dihydrochloride (intermediate A) (100 mg, 0.25 mmol) and 6-methyl-nicotinic acid.

Provenance & Evidence