4-(Propan-2-yl)benzene-1,2-diamine → HCID 178438824, compound

HRID 1424162Notes

Reaction equation

HRID 1424162 reaction equation
C(OC([N:8]1[C@H:12]([C:13](O)=O)[C@@H:11]([CH:16]([CH3:18])[CH3:17])[O:10]C1(C)C)=O)(C)(C)C.[CH3:21][CH:22]([C:24]1[CH:25]=[C:26]([NH2:31])[C:27]([NH2:30])=[CH:28][CH:29]=1)[CH3:23]>>[NH2:8][C@H:12]([C:13]1[NH:30][C:27]2[CH:28]=[CH:29][C:24]([CH:22]([CH3:21])[CH3:23])=[CH:25][C:26]=2[N:31]=1)[C@H:11]([OH:10])[CH:16]([CH3:18])[CH3:17]

Participants

3

Reactant 2

HCID 50970284-(Propan-2-yl)benzene-1,2-diamineHCID 70021709(4S,5R)-3-(tert-butoxycarbonyl)-5-isopropyl-2,2-dimethyl-1,3-oxazolidine-4-carboxylic acid

Product 1

HCID 178438824HCID 178438824, compound

Procedure

The title compound was prepared according to Method 4 using (4S,5R)-3-(tert-butoxycarbonyl)-5-isopropyl-2,2-dimethyl-1,3-oxazolidine-4-carboxylic acid (Preparation 60) and 4-(1-methylethyl)-1,2-benzenediamine.

Sources & evidence

ORD record
ord-a591b94cc0e546e79401971555f9e99d
Source dataset
uspto-grants-2015_01
Patent number
US08927587B2

Reaction notes

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